Antibiotic (Penicillin)
Brand of Procaine Penicillin, Benzyl Penicillin Potassium
Last reviewed June 2026
Who is this for?
This is a combination antibiotic injection that contains two forms of penicillin — Procaine Penicillin (which releases slowly and lasts longer in the body) and Benzyl Penicillin Potassium (which works fast to kill bacteria quickly). Together, they give you both immediate and long-lasting protection against bacterial infections.
Inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins and preventing peptidoglycan cross-linking, resulting in bactericidal activity against susceptible Gram-positive and Gram-negative organisms.
Prescription Required
You need a doctor's prescription to buy this drug.
Explore this drug
This drug is given as an injection into the muscle (IM injection) by a nurse or doctor — it is NOT taken by mouth. Adults typically receive 1 to 4 mega units (million units) daily, depending on how serious the infection is. Your doctor will decide the exact dose and how many days you need it. Always complete the full course even if you feel better.
If you miss your scheduled injection, go to the hospital or clinic as soon as you remember. Do not try to double the dose. Contact your doctor to reschedule and continue the remaining doses as planned.
Important for antibiotics
Always complete the full course even if you feel better. Stopping early can cause the infection to return and become drug-resistant.
Methotrexate (used for arthritis and some cancers) — penicillin can increase its side effects. Blood-thinning drugs like warfarin — penicillin may increase the risk of bleeding. Tetracycline antibiotics (like doxycycline) — taking them together can reduce how well penicillin works, so tell your doctor about any other medications you are using.
Check your specific combination
Is it safe to take Procaine with your other drugs?
Penicillin is generally considered safe during pregnancy and breastfeeding, but always inform your doctor that you are pregnant or breastfeeding before receiving this injection.
Store the powdered form in a cool, dry place away from direct sunlight and heat — Nigerian weather can be very hot, so avoid storing near windows or in cars. Once mixed with water for injection, use it immediately or refrigerate and use within 24 hours. Always keep out of reach of children.
For information only — not medical advice. Always talk to a doctor or pharmacist before changing your medication.
Names this drug is sold under — especially in Nigerian and West African pharmacies
Counterfeit Drug Warning
Fake drugs are a serious problem in Nigeria. Always buy from a registered pharmacy. If the packaging looks different from what is described above, do not use it.
Genuine packaging for Caine Pen Injection 4 Mega
Packaging image coming soon
We're building our packaging database — check back soon
NAFDAC Number
A4-3033
Verify Your Pack